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泛托法隆Fantofarone 是钙离子通道 (Calcium Channel) 的强效拮抗剂。
物化属性:
密度:1.16
熔点:82-83°
折射率:1.573
PSA:77.86000
LOGP:6.93690
[1]. Adovelande J, et al. Synergy between two calcium channel blockers, verapamil and fantofarone (SR33557), in reversing chloroquine resistance in Plasmodium falciparum. Biochem Pharmacol. 1998 Feb 15;55(4):433-40.
[2]. Dongay B, et al. Effect of fantofarone, a new Ca2+ channel antagonist, on angioplasty-induced vasospasm in an atherosclerotic rabbit model. Biochem Pharmacol. 1998 Jun 15;55(12):2047-50.
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