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SR9011 是一种 REV-ERBα/β 激动剂,作用于 REV-ERBα 和 REV-ERBβ,IC50s 分别为 790 nM 和 560 nM。
[1]. Solt LA, et al. Regulation of circadian behaviour and metabolism by synthetic REV-ERB agonists. Nature. 2012 Mar 29;485(7396):62-8.
[2]. Wang Y, et al. Anti-proliferative actions of a synthetic REV-ERBα/β agonist in breast cancer cells. Biochem Pharmacol. 2015 Aug 15;96(4):315-22.
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