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1A-116 是一种特异性 Rac1 抑制剂。
物化属性:
密度:1.22±0.1 g/cm3(Predicted)
沸点:357.5±52.0 °C(Predicted)
[1]. Gonzalez N, et al. Pharmacological inhibition of Rac1-PAK1 axis restores tamoxifen sensitivity in human resistant breast cancer cells. Cell Signal. 2017 Jan;30:154-161.
[2]. Cardama GA, et al. Preclinical development of novel Rac1-GEF signaling inhibitors using a rational design approach in highly aggressive breast cancer cell lines. Anticancer Agents Med Chem. 2014;14(6):840-51.
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