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产品描述:
Clevidipine Butyrate是一种二氢吡啶类钙离子通道抑制剂,用于降血压。
靶点:
Calcium channel
中文别名:
丁酸氯维地平;
4-(2,3-二氯苯基)-1,4-二氢-2,6-二甲基-3,5-吡啶二甲酸甲基(1-丁酰氧基)甲酯
物化属性:
密度:1.289
熔点:128-130°C
沸点:539.7°C at 760 mmHg
折射率:1.542
闪光点:280℃
[1]. Yi X, Vivien B, Lynch C 3rd. Clevidipine blockade of L-type Ca2+ currents: steady-state and kinetic electrophysiological studies in guinea pigventricular myocytes.
[2]. Huraux C, Makita T, Szlam F, The vasodilator effects of clevidipine on human internal mammary artery. Anesth Analg. 1997 Nov;85(5):1000-4.
[3]. Ericsson H, et al. In vitro hydrolysis rate and protein binding of clevidipine, a new ultrashort-acting calcium antagonist metabolised by esterases, in different animal species and man. Eur J Pharm Sci. 1999 Apr;8(1):29-37.
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