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产品描述:
醋酸亮丙瑞林 Leuprolide acetate 是一种合成的九肽,是GnRHR的激动剂,用于多种临床治疗,包括前列腺癌、子宫内膜异位、子宫平滑肌瘤、中枢性性早熟和体外受精。
中文别名:
醋酸亮丙瑞林, 一种垂体促性腺激素受体抑制剂
物化属性:
外观与形状:松软的固体
密度:1.44
熔点:150-155°C
沸点:1720.5°C at 760 mmHg
折射率:1.681
闪光点:994.3°C
PSA:466.34000
LOGP:3.44730
[1]. Mizutani T, Sugihara A, Nakamuro K, Suppression of cell proliferation and induction of apoptosis in uterine leiomyoma by gonadotropin-releasing hormone agonist (leuprolide acetate). J Clin Endocrinol Metab. 1998 Apr;83(4):1253-5.
[2]. Silva AL, Abreu LG, Rosa-e-Silva AC, Leuprolide acetate reduces both in vivo and in vitro ovarian steroidogenesis in infertile women undergoing assisted reproduction. Steroids. 2008 Dec 22;73(14):1475-84.
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