0576-88813233
GNF-2是非ATP竞争性的Bcr-Abl选择性抑制剂,IC50为140nM。
中文名称:
3-[6-[[4-(三氟甲氧基)苯基]氨基]-4-嘧啶基]苯甲酰胺
物化属性:
密度:1.405
沸点:536.4°C at 760 mmHg
折射率:1.611
闪光点:278.2°C
PSA:90.13000
LOGP:4.65800
[1]. Adrián FJ, et al. Allosteric inhibitors of Bcr-abl-dependent cell proliferation. Nat Chem Biol. 2006 Feb;2(2):95-102.
[2]. Khateb M, et al. Overcoming Bcr-Abl T315I mutation by combination of GNF-2 and ATP competitors in an Abl-independent mechanism. BMC Cancer. 2012 Nov 27;12:563.
版权所有 Copyright(C) 2018-2022 台州市科瑞生物技术有限公司